SCHEMBL19780167

SCHEMBL19780167

COc1cc2c(C)n[nH]c2cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 3/20 0.49
GABRD O14764 3/20 0.49
GABRA1 P14867 3/20 0.49
GABRB1 P18505 3/20 0.49
GABRG2 P18507 3/20 0.49
GABRB3 P28472 3/20 0.49
GABRA5 P31644 3/20 0.49
GABRA3 P34903 3/20 0.49
GABRA2 P47869 3/20 0.49
GABRB2 P47870 3/20 0.49
GABRA4 P48169 3/20 0.49
GABRE P78334 3/20 0.49
GABRA6 Q16445 3/20 0.49
GABRG1 Q8N1C3 3/20 0.49
GABRG3 Q99928 3/20 0.49
GABRQ Q9UN88 3/20 0.49
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
LRRK2 Q5S007 1/20 0.39
DYRK1A Q13627 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16517816 0.81 GABRP (0.47) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL25862554 0.78 DYRK1A (0.39) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL13906113 0.78 ADORA2A (0.44) ADORA2AADORA2BDYRK1APIM1MAP2K4
SCHEMBL7920977 0.77 ADORA2A (0.47) ADORA2AADORA2BDYRK1APIM1
SCHEMBL16517106 0.76 PRKAG1 (0.53) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL16516994 0.74 KDM4E (0.54) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL24121819 0.74 ADORA2A (0.44) ADORA2AADORA2BDYRK1APIM1MAP2K4
SCHEMBL19965414 0.74 ADORA2A (0.44) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL17514109 0.72 GABRA1 (0.55) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL17683153 0.72 ADORA2A (0.50) ADORA2AADORA2BCHEK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018011628-A1 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2018-01-18 WO disclosed