SCHEMBL19781860

SCHEMBL19781860

CCCn1cc(C#N)cn1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.47
KCNJ5 P48544 3/20 0.41
IRAK4 Q9NWZ3 3/20 0.39
CYP11B2 P19099 3/20 0.38
CYP19A1 P11511 1/20 0.36
PIK3CD O00329 1/20 0.35
PIP5K1C O60331 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PI4KA P42356 1/20 0.35
PIK3CG P48736 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
AR P10275 2/20 0.34
PGR P06401 1/20 0.34
ADORA2B P29275 1/20 0.34
NLRP3 Q96P20 1/20 0.34
EP300 Q09472 1/20 0.34
CREBBP Q92793 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18641909 0.89 L3MBTL1 (0.38) L3MBTL1KCNJ5IRAK4CYP11B2CYP19A1
SCHEMBL5796848 0.87 CYP19A1 (0.39) L3MBTL1KCNJ5CYP11B2CYP19A1
SCHEMBL7462189 0.84
SCHEMBL23174810 0.81 IRAK4 (0.39) IRAK4CYP11B2ARPGREP300
SCHEMBL1935296 0.81 CYP19A1 (0.34) CYP11B2CYP19A1ARPGRNLRP3
SCHEMBL25359893 0.81 L3MBTL1 (0.47) L3MBTL1KCNJ5IRAK4PIK3CDPIP5K1C
SCHEMBL25362235 0.77 L3MBTL1 (0.44) L3MBTL1KCNJ5PIK3CDPIP5K1CPIK3CA
SCHEMBL26962749 0.77 NLRP3 (0.39) L3MBTL1IRAK4CYP11B2CYP19A1AR
SCHEMBL10789578 0.76
SCHEMBL21265473 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013615-A1 C7, C12, AND C16 SUBSTITUTED NEUROACTIVE STEROIDS AND THEIR METHODS OF USE SAGE THERAPEUTICS, INC. (US) 2018-01-18 WO disclosed