SCHEMBL19782739

SCHEMBL19782739

Cc1cc(OCCNSc2ccc(F)cc2)cc2sc(Br)nc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2RL3 Q96RI0 3/20 0.34
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
MAPT P10636 3/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HTT P42858 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HTR7 P34969 4/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19783269 0.81 IKBKB (0.31)
SCHEMBL30189952 0.79 F2RL3 (0.51) F2RL3MAPTHTTTDP1TP53
SCHEMBL19782740 0.79 F2RL3 (0.51) F2RL3MAPTHTTTDP1TP53
SCHEMBL19783423 0.77 F2RL3 (0.54) F2RL3
SCHEMBL19782945 0.74 F2RL3 (0.52) F2RL3
SCHEMBL30189754 0.72 HSD17B10 (0.37) F2RL3MAPTNPC1RAB9AHTT
SCHEMBL19783059 0.72 HSD17B10 (0.37) F2RL3MAPTNPC1RAB9AHTT
SCHEMBL19783647 0.71 MAPT (0.44) MAPTNPC1RAB9ASMN1; SMN2HTT
SCHEMBL21395510 0.69 CA12 (0.45) HTTLMNACYP1A2CYP3A4CYP2C9
SCHEMBL30189776 0.69 CA12 (0.45) HTTLMNACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed