SCHEMBL19782767

SCHEMBL19782767

Nc1ccnc(OCCI)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 3/20 0.38
LOX P28300 2/20 0.38
ASIC3 Q9UHC3 1/20 0.36
NOS3 P29474 3/20 0.33
NOS1 P29475 3/20 0.33
NOS2 P35228 3/20 0.33
KDM4E B2RXH2 3/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
ALDH1A1 P00352 3/20 0.33
GAA P10253 3/20 0.33
MAPT P10636 3/20 0.33
TP53 P04637 2/20 0.33
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
CASP1 P29466 1/20 0.33
HTT P42858 1/20 0.33
CASP7 P55210 1/20 0.33
ATM Q13315 1/20 0.33
NUDT1 P36639 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340745 0.82 MAPT (0.50) LOXL2LOXASIC3NOS3NOS1
SCHEMBL2144434 0.82 LOXL2 (0.43) LOXL2LOXASIC3NOS3NOS1
SCHEMBL4101483 0.81 TSHR (0.46) LOXL2LOXKDM4EMEN1KMT2A
SCHEMBL27854114 0.81 LOXL2 (0.38) LOXL2LOXASIC3NOS3NOS1
SCHEMBL5323724 0.81 LOX (0.42) LOXL2LOXASIC3NOS3NOS1
SCHEMBL23462840 0.81 ASIC3 (0.40) LOXL2LOXASIC3NOS3NOS1
SCHEMBL16265338 0.81 LOXL2 (0.42) LOXL2LOXASIC3NOS3NOS1
SCHEMBL940535 0.78 HTR7 (0.46) MAPT
SCHEMBL171947 0.78 TP53 (0.48) LOXL2LOXASIC3NOS3NOS1
SCHEMBL29218081 0.76 LOXL2 (0.40) LOXL2LOXASIC3NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed