SCHEMBL19782949

SCHEMBL19782949

O=Cc1cc(O)cc2sc(Br)nc12

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.34
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
HSD17B1 P14061 1/20 0.33
NSD1 Q96L73 1/20 0.33
DYRK1A Q13627 1/20 0.33
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395529 0.76 ERN1 (0.39) ERN1DYRK1AHTT
SCHEMBL19782753 0.73 HSD17B10 (0.42) ESR1ESR2NSD1DYRK1AGAA
SCHEMBL19782540 0.73 ALDH1A1 (0.42) HSD17B1NSD1GAAHTT
SCHEMBL30189617 0.73 ALDH1A1 (0.42) HSD17B1NSD1GAAHTT
SCHEMBL20305619 0.69 ALOX5 (0.46) DYRK1AGAAHTT
SCHEMBL19782536 0.68 NSD1 (0.33) ESR1ESR2NSD1
SCHEMBL2274086 0.66 RAB9A (0.39) GAAHTT
SCHEMBL25612184 0.64 ERN1 (0.43) ERN1ESR1ESR2
SCHEMBL1360479 0.64 HTT (0.63) HSD17B1DYRK1AGAAHTTL3MBTL1
SCHEMBL21379622 0.64 APP (0.37) DYRK1AGAAHTTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed