SCHEMBL19785912

SCHEMBL19785912

CCc1nnc(Nc2cc(C)cc(CN3CCNCC3)c2C)o1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FASN P49327 1/20 0.36
LMNA P02545 1/20 0.34
SOS1 Q07889 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
KDM1A O60341 1/20 0.31
CXCR4 P61073 1/20 0.30
CYP1A2 P05177 1/20 0.30
CHRM2 P08172 1/20 0.30
SLC6A4 P31645 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19785916 0.82 LMNA (0.33) LMNA
SCHEMBL22383769 0.79 SMN1; SMN2 (0.39) FASN
SCHEMBL22383768 0.79 FASN (0.36) FASN
SCHEMBL19785619 0.79 SMN1; SMN2 (0.40) FASNLMNA
SCHEMBL21368556 0.70 XIAP (0.32)
SCHEMBL22430963 0.70 XIAP (0.36)
SCHEMBL19785915 0.70 XIAP (0.32)
Hydrochloric Acid SCHEMBL21354282 0.70 XIAP (0.32)
Hydrochloric Acid SCHEMBL21354250 0.70 XIAP (0.32)
Hydrochloric Acid SCHEMBL21354290 0.70 XIAP (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484880-B1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA AS (DK) 2020-09-02 EP disclosed
WO-2018011201-A1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2018-01-18 WO disclosed