SCHEMBL1979037

SCHEMBL1979037

CCN(CC)CCOc1ccc(-c2c(OC)ccc3[nH]c4cnc(-c5cccnc5)cc4c23)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 1/20 0.48
ABL1 P00519 1/20 0.46
BCR P11274 1/20 0.46
PIM1 P11309 2/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
KDR P35968 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CDK2AP1 O14519 1/20 0.38
CHEK1 O14757 1/20 0.38
MCHR1 Q99705 1/20 0.38
LYN P07948 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980602 0.92 ABL1 (0.45) NEK1ABL1BCRPIM1PIM3
SCHEMBL1979625 0.85 TLR8 (0.45) NEK1ABL1BCRPIM1PIM3
SCHEMBL1980257 0.84 PIM1 (0.52) PIM1PIM3PIM2TLR8TLR7
SCHEMBL1983423 0.84 ABL1 (0.47) ABL1BCRPIM1TLR8TLR7
SCHEMBL2214322 0.82 PIM1 (0.40) ABL1BCRPIM1PIM3PIM2
SCHEMBL1980317 0.82 PDPK1 (0.49) ABL1BCRTLR8TLR7CYP2D6
SCHEMBL1979697 0.82 TLR8 (0.40) NEK1PIM1PIM3PIM2TLR8
SCHEMBL1984174 0.82 ABL1 (0.49) ABL1BCRNPC1RAB9A
SCHEMBL1979485 0.81 ABL1 (0.49) ABL1BCRTLR8TLR7KDR
SCHEMBL12597452 0.81 PIM1 (0.49) PIM1PIM3PIM2TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed