SCHEMBL1979485

SCHEMBL1979485

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(OCCCN2CCOCC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.49
BCR P11274 2/20 0.49
KDR P35968 1/20 0.43
PADI4 Q9UM07 1/20 0.42
HRH3 Q9Y5N1 2/20 0.42
PDPK1 O15530 1/20 0.42
EPHX2 P34913 1/20 0.41
CYP2D6 P10635 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
JAK3 P52333 1/20 0.41
MAPK9 P45984 4/20 0.40
MAPKAPK2 P49137 4/20 0.40
UBE2N P61088 1/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
CHEK1 O14757 1/20 0.40
ACHE P22303 1/20 0.40
AVPR1B P47901 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1984174 0.96 ABL1 (0.49) ABL1BCRPADI4MAPK9MAPKAPK2
SCHEMBL1980317 0.92 PDPK1 (0.49) ABL1BCRHRH3PDPK1CYP2D6
SCHEMBL1983423 0.89 ABL1 (0.47) ABL1BCRKDRPDPK1TLR8
SCHEMBL1979784 0.87 PKM (0.47)
SCHEMBL1984242 0.85 EPHX2 (0.46) ABL1BCRPADI4HRH3EPHX2
SCHEMBL1980602 0.82 ABL1 (0.45) ABL1BCRTLR8TLR7
SCHEMBL1980375 0.82 JAK2 (0.45) ABL1BCRJAK2JAK1JAK3
SCHEMBL1979037 0.81 NEK1 (0.48) ABL1BCRKDRCYP2D6TLR8
SCHEMBL1561132 0.81 PADI4 (0.47) ABL1BCRPADI4EPHX2CYP2D6
SCHEMBL2217947 0.80 CHEK1 (0.62) ABL1BCRHRH3EPHX2CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO claimed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed