SCHEMBL1979697

SCHEMBL1979697

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(OCC(C)CN(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.40
TLR7 Q9NYK1 2/20 0.40
PIM1 P11309 7/20 0.39
PIM3 Q86V86 3/20 0.39
PIM2 Q9P1W9 3/20 0.39
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
NEK1 Q96PY6 1/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
NPY5R Q15761 1/20 0.35
DYRK1A Q13627 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HSD17B10 Q99714 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
CLK4 Q9HAZ1 3/20 0.35
CLK2 P49760 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980602 0.87 ABL1 (0.45) TLR8TLR7PIM1PIM3PIM2
SCHEMBL1560888 0.83 PIM1 (0.39) PIM1PIM3PIM2NPC1RAB9A
SCHEMBL12597224 0.83 PTAFR (0.44) TLR8TLR7DYRK1AALDH1A1
SCHEMBL1980257 0.82 PIM1 (0.52) TLR8TLR7PIM1PIM3PIM2
SCHEMBL1979037 0.82 NEK1 (0.48) TLR8TLR7PIM1PIM3PIM2
SCHEMBL12597452 0.80 PIM1 (0.49) TLR8TLR7PIM1PIM3PIM2
SCHEMBL1978448 0.79 PIM1 (0.45) TLR8TLR7PIM1PIM3PIM2
SCHEMBL1983423 0.79 ABL1 (0.47) TLR8TLR7PIM1DYRK1ACLK2
SCHEMBL1979784 0.79 PKM (0.47) ALDH1A1KDM4E
SCHEMBL12597231 0.79 NEK1 (0.52) TLR8TLR7PIM1PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed