SCHEMBL1980602

SCHEMBL1980602

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(OCCN(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.45
BCR P11274 2/20 0.45
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
PIM1 P11309 3/20 0.41
PIM3 Q86V86 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
NEK1 Q96PY6 2/20 0.41
CLK2 P49760 1/20 0.40
DYRK1A Q13627 1/20 0.40
ITGA4 P13612 1/20 0.40
NAPEPLD Q6IQ20 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
WNT1 P04628 1/20 0.39
TGFBR1 P36897 1/20 0.39
PAX8 Q06710 1/20 0.39
TLR8 Q9NR97 2/20 0.39
TLR7 Q9NYK1 2/20 0.39
HCRTR1 O43613 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979037 0.92 NEK1 (0.48) ABL1BCRPIM1PIM3PIM2
SCHEMBL1979697 0.87 TLR8 (0.40) PIM1PIM3PIM2NEK1CLK2
SCHEMBL1980257 0.85 PIM1 (0.52) PIM1PIM3PIM2CLK2DYRK1A
SCHEMBL1983423 0.85 ABL1 (0.47) ABL1BCRCHRNB2CHRNA4PIM1
SCHEMBL1982709 0.84 TLR8 (0.48) ABL1BCRPIM1PIM3PIM2
SCHEMBL1981277 0.84 WNT1 (0.49) ABL1BCRDYRK1AWNT1TLR8
SCHEMBL1980317 0.84 PDPK1 (0.49) ABL1BCRTLR8TLR7
SCHEMBL1980014 0.84 TLR7 (0.49) ABL1BCRPIM1PIM3PIM2
SCHEMBL1984174 0.83 ABL1 (0.49) ABL1BCRNPC1RAB9ATGFBR1
SCHEMBL1978130 0.82 TLR7 (0.48) ABL1BCRDYRK1AWNT1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed