SCHEMBL7958615

SCHEMBL7958615

CCCCCCCC1CC2(NC(=O)NC2=O)c2cc(Br)ccc2O1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 0.43
AKR1B10 O60218 2/20 0.43
AKR1A1 P14550 2/20 0.43
SIRT2 Q8IXJ6 1/20 0.36
CYP1A2 P05177 2/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7957154 0.90 SIRT2 (0.35) AKR1B1AKR1B10AKR1A1SIRT2CYP1A2
SCHEMBL10579227 0.88 AKR1B1 (0.43) AKR1B1AKR1B10AKR1A1
SCHEMBL10576515 0.86 AKR1B1 (0.59) AKR1B1AKR1B10AKR1A1SIRT2MAPT
SCHEMBL10573588 0.83 AKR1B1 (0.45) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL1979448 0.80 AKR1B1 (0.45) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10575201 0.78 AKR1B1 (0.47) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10571505 0.78 AKR1B1 (0.62) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL1978738 0.74 AKR1B1 (0.48) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL9836968 0.74 AKR1B1 (0.62) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10574757 0.73 AKR1B1 (0.65) AKR1B1AKR1B10AKR1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed