SCHEMBL1979835

SCHEMBL1979835

CC(C)CCC#Cc1c[c]ccc1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.35
SIGMAR1 Q99720 1/20 0.32
GRM5 P41594 1/20 0.31
CHRNB2 P17787 3/20 0.30
CHRNA4 P43681 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL614112 0.84 HRH3 (0.38) HTR2ACHRNB2CHRNA4
SCHEMBL1978631 0.83 HTR2A (0.44) HTR2ASIGMAR1
SCHEMBL8130889 0.78 HTR2A (0.55) HTR2ASIGMAR1GRM5
SCHEMBL614587 0.78 KCNH2 (0.39) CHRNB2CHRNA4
SCHEMBL482776 0.77 NPSR1 (0.39) HTR2ACHRNB2CHRNA4
SCHEMBL8114656 0.75 KCNH2 (0.47)
SCHEMBL8122306 0.75 KCNH2 (0.47)
SCHEMBL8122540 0.75 KCNH2 (0.47)
SCHEMBL6293461 0.74 CHRNB2 (0.50) HTR2ASIGMAR1CHRNB2CHRNA4
SCHEMBL1984212 0.73 HAO1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO claimed
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed