SCHEMBL1979899

SCHEMBL1979899

CCOC(=O)c1cnc(N)n1C

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 5/20 0.49
KDM4E B2RXH2 3/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
IDO1 P14902 4/20 0.43
MAPT P10636 2/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HSP90AA1 P07900 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11773323 0.98 CSNK1D (0.48) CSNK1DKDM4ENPC1RAB9AALDH1A1
SCHEMBL28720076 0.83 IDO1 (0.45) KDM4ENPC1RAB9AALDH1A1KMT2A
SCHEMBL8700542 0.81 SMN1; SMN2 (0.48) KDM4ENPC1RAB9AALDH1A1MEN1
SCHEMBL998243 0.80 IDO1 (0.43) KDM4ENPC1RAB9AKMT2AIDO1
SCHEMBL28616856 0.80 IDO1 (0.47) KDM4ENPC1RAB9AALDH1A1KMT2A
SCHEMBL23108117 0.80 CSNK1D (0.49) CSNK1DKDM4ENPC1RAB9AALDH1A1
SCHEMBL26354914 0.78 IDO1 (0.41) CSNK1DKDM4ENPC1RAB9AKMT2A
SCHEMBL12381781 0.78 SMN1; SMN2 (0.52) KDM4ENPC1RAB9AALDH1A1MEN1
SCHEMBL11961046 0.78 ADORA3 (0.44) KDM4ENPC1RAB9AALDH1A1MEN1
SCHEMBL23108232 0.77 GRK6 (0.47) CSNK1DKDM4ENPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240425461-A1 PREPARATION PROCESS OF INTERMEDIATE, SYNTHESIS PROCESS OF AMINO IMIDAZOLE CARBOXYLATE ESTER AND HPLC PURITY MEASURE METHOD ASCENTAWITS PHARMACEUTICALS, LTD. (CN) 2024-12-26 US claimed
CN-116789558-A Preparation method of intermediate, synthesis method of amino imidazole carboxylate and HPLC (high performance liquid chromatography) purity detection method 深圳艾欣达伟医药科技有限公司 2023-09-22 CN claimed
US-20240425462-A1 Preparation Process of 1-N-Methyl-2-Nitro-5-Hydroxymethyl Imidazole ASCENTAWITS PHARMACEUTICALS, LTD. (CN) 2024-12-26 US disclosed
US-20240425461-A1 PREPARATION PROCESS OF INTERMEDIATE, SYNTHESIS PROCESS OF AMINO IMIDAZOLE CARBOXYLATE ESTER AND HPLC PURITY MEASURE METHOD ASCENTAWITS PHARMACEUTICALS, LTD. (CN) 2024-12-26 US disclosed
US-20240343710-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF 1CBIO, INC. 2024-10-17 US disclosed
US-12115226-B2 Linker containing arylnitro, antibody-drug conjugate containing linker and use of linker ACADEMY OF MILITARY MEDICAL SCIENCES (CN) 2024-10-15 US disclosed
WO-2024178127-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF 1CBIO, INC. (US) 2024-08-29 WO disclosed
US-20230303618-A1 TRIPTOLIDE CONJUGATES AND USES THEREOF REYOUNG CORPORATION (US) 2023-09-28 US disclosed
CN-116803989-A Preparation process of 1-N-methyl-2-nitro-5-hydroxymethyl imidazole 深圳艾欣达伟医药科技有限公司 2023-09-26 CN disclosed
CN-116789558-A Preparation method of intermediate, synthesis method of amino imidazole carboxylate and HPLC (high performance liquid chromatography) purity detection method 深圳艾欣达伟医药科技有限公司 2023-09-22 CN disclosed
CN-112601556-B Linker containing aromatic nitro group, antibody conjugate drug containing linker and application of linker 中国人民解放军军事科学院军事医学研究院 2022-08-09 CN disclosed
US-7550496-B2 Compositions and methods for treating cancer THRESHOLD PHARMACEUTICALS, INC. (US) 2009-06-23 US disclosed
EP-1896040-A2 PHOSPHORAMIDATE ALKYLATOR PRODRUGS Threshold Pharmaceuticals, Inc. (US) 2008-03-12 EP disclosed
WO-2007002931-A2 PHOSPHORAMIDATE ALKYLATOR PRODRUGS THRESHOLD PHARMACEUTICALS, INC. (US) 2007-01-04 WO disclosed
WO-2007002931-A2 PHOSPHORAMIDATE ALKYLATOR PRODRUGS THRESHOLD PHARMACEUTICALS, INC. (US) 2007-01-04 WO disclosed
US-5843942-A Aromatic amino ethers as pain relieving agents ZENECA LIMITED (GB) 1998-12-01 US disclosed
EP-0773930-A1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LIMITED (GB) 1997-05-21 EP disclosed
WO-1996003380-A1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LIMITED (GB) 1996-02-08 WO disclosed
US-3987053-A ANTIMICROBIAL GRUPPO LEPETIT S.P.A. (IT) 1976-10-19 US disclosed
US-3954789-A 2-Nitroimidazole derivatives GRUPPO LEPETIT S.P.A. (IT) 1976-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240343710-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF PARP1, PARP11, PARP12 CSNK1D 673/4885KDM4E 1701/4885NPC1 2461/4885
US-20240425462-A1 Preparation Process of 1-N-Methyl-2-Nitro-5-Hydroxymethyl Imidazole DNMT1, COX4I1, NDC1 CSNK1D 516/4885KDM4E 612/4885NPC1 662/4885
US-20240425461-A1 PREPARATION PROCESS OF INTERMEDIATE, SYNTHESIS PROCESS OF AMINO IMIDAZOLE CARBOXYLATE ESTER AND HPLC PURITY MEASURE METHOD ABAT, ALDH7A1, IDH2 CSNK1D 1582/4885KDM4E 260/4885NPC1 4246/4885
US-12115226-B2 Linker containing arylnitro, antibody-drug conjugate containing linker and use of linker BCR, FCGR2A, FCGRT CSNK1D 2892/4885KDM4E 2409/4885NPC1 1422/4885
US-20230303618-A1 TRIPTOLIDE CONJUGATES AND USES THEREOF TLR9, XIAP, ENPP2 CSNK1D 2640/4885KDM4E 2714/4885NPC1 2162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.