SCHEMBL1980342

SCHEMBL1980342

CCCCN(Cc1c(Cl)cccc1Cl)c1nnc(-c2cc(C)c(OC)c(C)c2)s1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 18/20 0.47
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
UBE2N P61088 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
S1PR3 Q99500 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981001 0.89 S1PR1 (0.46) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1981553 0.88 S1PR1 (0.51) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1981536 0.85 S1PR1 (0.52) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1984811 0.83 S1PR1 (0.49) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1979699 0.83 CPB1 (0.39) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1981126 0.81 S1PR1 (0.50) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1980288 0.81 S1PR1 (0.41) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1980417 0.81 S1PR1 (0.50) S1PR1ALDH1A1S1PR3
SCHEMBL1982705 0.80 S1PR1 (0.43) S1PR1KDM4EALDH1A1HPGDUBE2N
SCHEMBL1967413 0.80 KDM4E (0.57) S1PR1KDM4EALDH1A1HPGDUBE2N

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP claimed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed
WO-2011069647-A1 NEW 2-AMINOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-06-16 WO disclosed