SCHEMBL1980288

SCHEMBL1980288

CCCCN(Cc1ccccc1C#N)c1nnc(-c2cc(C)c(OC)c(C)c2)s1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 12/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
HSD17B10 Q99714 3/20 0.40
HPGD P15428 2/20 0.40
UBE2N P61088 1/20 0.40
LMNA P02545 1/20 0.38
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
CPB1 P15086 1/20 0.35
USP2 O75604 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
POLB P06746 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12600003 0.89 S1PR1 (0.43) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981001 0.86 S1PR1 (0.46) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981126 0.86 S1PR1 (0.50) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981536 0.83 S1PR1 (0.52) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL2230853 0.82 S1PR1 (0.49) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1980342 0.81 S1PR1 (0.47) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1979699 0.80 CPB1 (0.39) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1982705 0.79 S1PR1 (0.43) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981553 0.79 S1PR1 (0.51) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1984811 0.78 S1PR1 (0.49) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP claimed
WO-2011069647-A1 NEW 2-AMINOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-06-16 WO claimed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed
WO-2011069647-A1 NEW 2-AMINOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-06-16 WO disclosed