SCHEMBL1980659

SCHEMBL1980659

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(C(=O)NCC(C)(C)CN(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 3/20 0.39
TLR8 Q9NR97 2/20 0.39
SMPD1 P17405 1/20 0.38
PTAFR P25105 1/20 0.38
TLR9 Q9NR96 1/20 0.38
IGF1R P08069 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
ALDH1A1 P00352 2/20 0.37
USP2 O75604 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HPSE Q9Y251 1/20 0.36
WNT1 P04628 1/20 0.36
DYRK1A Q13627 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 1/20 0.36
BLM P54132 1/20 0.36
ABL1 P00519 3/20 0.36
BCR P11274 3/20 0.36
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981277 0.88 WNT1 (0.49) TLR7TLR8SMPD1PTAFRTLR9
SCHEMBL1978130 0.87 TLR7 (0.48) TLR7TLR8PTAFRTLR9L3MBTL1
SCHEMBL1979456 0.86 PTAFR (0.47) TLR7TLR8PTAFRTLR9L3MBTL1
SCHEMBL1981901 0.85 CHEK1 (0.40) TLR7TLR8SMPD1PTAFRTLR9
SCHEMBL1983761 0.85 BRAF (0.47) TLR7SMPD1PTAFRTLR9L3MBTL1
SCHEMBL1981803 0.85 MTNR1A (0.45) TLR7TLR8SMPD1PTAFRTLR9
SCHEMBL473735 0.84 CHEK1 (0.39) WNT1DYRK1APIM1PIM3PIM2
SCHEMBL1981315 0.84 PTAFR (0.47) TLR7SMPD1PTAFRTLR9ALDH1A1
SCHEMBL12597224 0.84 PTAFR (0.44) TLR7TLR8SMPD1PTAFRTLR9
SCHEMBL12598112 0.83 TLR7 (0.45) TLR7TLR8SMPD1PTAFRTLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed