SCHEMBL19807679

SCHEMBL19807679

FC(F)(F)c1ncc(-n2cc(CCl)c(C(F)(F)F)n2)cn1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 12/20 0.43
FGFR1 P11362 1/20 0.43
DGAT1 O75907 2/20 0.33
MPO P05164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21010418 0.84 TRPA1 (0.43) TRPA1FGFR1DGAT1MPO
SCHEMBL19807684 0.84 TRPA1 (0.45) TRPA1FGFR1DGAT1
SCHEMBL20997476 0.84 TRPA1 (0.45) TRPA1FGFR1DGAT1
SCHEMBL19807681 0.81 TRPA1 (0.41) TRPA1FGFR1MPO
SCHEMBL17979414 0.80 TRPA1 (0.46) TRPA1FGFR1
SCHEMBL19807437 0.80 TRPA1 (0.52) TRPA1FGFR1DGAT1
SCHEMBL18017677 0.77 TRPA1 (0.46) TRPA1FGFR1DGAT1
SCHEMBL19795020 0.77 TRPA1 (0.39) TRPA1FGFR1DGAT1
SCHEMBL19795019 0.72 PTGS2 (0.37) TRPA1FGFR1DGAT1
SCHEMBL3332657 0.69 POLB (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10766878-B2 Sulfonylcycloalkyl carboxamide compounds GENENTECH, INC. (US) 2020-09-08 US disclosed
US-20190144430-A1 SULFONYLCYCLOALKYL CARBOXAMIDE COMPOUNDS GENENTECH, INC. (US) 2019-05-16 US disclosed
WO-2018015411-A1 SULFONYLCYCLOALKYL CARBOXAMIDE COMPOUNDS AS TRPA1 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2018-01-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190144430-A1 SULFONYLCYCLOALKYL CARBOXAMIDE COMPOUNDS TRPA1, TRPV1, TRPV5 TRPA1 1/4885FGFR1 315/4885DGAT1 1478/4885
US-10766878-B2 Sulfonylcycloalkyl carboxamide compounds TRPA1, TRPV1, TRPV5 TRPA1 1/4885FGFR1 315/4885DGAT1 1478/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.