Lysine

Lysine

SCHEMBL1983160

NCCCCC(N)C(=O)O.O=C(O)c1nccs1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.56
ARG1 P05089 4/20 0.41
ALDH1A1 P00352 1/20 0.39
GRIK1 P39086 1/20 0.38
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
GRIK2 Q13002 1/20 0.38
GRIK3 Q13003 1/20 0.38
GRIK4 Q16099 1/20 0.38
GRIK5 Q16478 1/20 0.38
PLA2G4A P47712 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
ARG2 P78540 4/20 0.37
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL358312 1.00 GSR (0.56) GSRARG1ALDH1A1GRIK1GRIA1
SCHEMBL7375810 0.84 GSR (0.43) GSRALDH1A1PLA2G4ACES1
Serine SCHEMBL359195 0.81 ALDH1A1 (0.44) ARG1ALDH1A1GRIK1GRIA1GRIA2
Serine SCHEMBL359193 0.81 ALDH1A1 (0.44) ARG1ALDH1A1GRIK1GRIA1GRIA2
Cysteine SCHEMBL357652 0.80 PTGS1 (0.50) ARG1ALDH1A1GRIK1GRIA1GRIA2
SCHEMBL28096157 0.80 ALDH1A1 (0.47) ALDH1A1PLA2G4ACES1
Cysteine SCHEMBL1986796 0.80 PTGS1 (0.50) ARG1ALDH1A1GRIK1GRIA1GRIA2
SCHEMBL7377556 0.80 ALDH1A1 (0.43) GSRARG1ALDH1A1GRIK1GRIA1
SCHEMBL358313 0.78 GSR (0.38) GSRALDH1A1PLA2G4ACES1
Glycine SCHEMBL359024 0.75 ALDH1A1 (0.52) ALDH1A1PLA2G4ACES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11992518-B2 Molecular vaccines for infectious disease AGILENT TECHNOLOGIES, INC. (US) 2024-05-28 US disclosed
US-10968269-B1 MHC multimers in borrelia diagnostics and disease AGILENT TECHNOLOGIES, INC. (US) 2021-04-06 US disclosed
US-20210047383-A1 MHC Multimers in Borrelia Diagnostics and Disease DAKO DENMARK APS (DK) 2021-02-18 US disclosed
US-20200347103-A1 MHC MULTIMERS IN TUBERCULOSIS DIAGNOSTICS, VACCINE AND THERAPEUTICS AGILENT TECHNOLOGIES INC (US) 2020-11-05 US disclosed
US-10611818-B2 MHC multimers in tuberculosis diagnostics, vaccine and therapeutics AGILENT TECHNOLOGIES, INC. (US) 2020-04-07 US disclosed
US-20190314471-A1 MOLECULAR VACCINES FOR INFECTIOUS DISEASE AGILENT TECHNOLOGIES, INC. 2019-10-17 US disclosed
US-10369204-B2 Molecular vaccines for infectious disease DAKO DENMARK A/S (DK) 2019-08-06 US disclosed
US-20120258126-A1 Molecular Vaccines for Infectious Disease DAKO DENMARK A/S (DK) 2012-10-11 US disclosed
US-20110318380-A1 MHC Multimers in Cancer Vaccines and Immune Monitoring DAKO DENMARK A/S (DK) 2011-12-29 US disclosed
US-20110236411-A1 MHC Multimers in Tuberculosis Diagnostics, Vaccine and Therapeutics DAKO DENMARK A/S (DE) 2011-09-29 US disclosed
EP-2337795-A2 MHC MULTIMERS IN CANCER VACCINES AND IMMUNE MONITORING Dako Denmark A/S (DK) 2011-06-29 EP disclosed
EP-2254592-A2 MHC MULTIMERS IN BORRELIA DIAGNOSTICS AND DISEASE Dako Denmark A/S (DK) 2010-12-01 EP disclosed
EP-2197908-A2 MHC MULTIMERS IN TUBERCULOSIS DIAGNOSTICS, VACCINE AND THERAPEUTICS Dako Denmark A/S (DK) 2010-06-23 EP disclosed
WO-2010037402-A1 MOLECULAR VACCINES FOR INFECTIOUS DISEASE DAKO DENMARK A/S (DK) 2010-04-08 WO disclosed
WO-2010037395-A2 MHC MULTIMERS IN CANCER VACCINES AND IMMUNE MONITORING DAKO DENMARK A/S (DK) 2010-04-08 WO disclosed
WO-2010037397-A1 MHC MULTIMERS IN CMV IMMUNE MONITORING DAKO DENMARK A/S (DK) 2010-04-08 WO disclosed
WO-2009106073-A2 MHC MULTIMERS IN BORRELIA DIAGNOSTICS AND DISEASE DAKO DENMARK A/S (DK) 2009-09-03 WO disclosed
WO-2009039854-A2 MHC MULTIMERS IN TUBERCULOSIS DIAGNOSTICS, VACCINE AND THERAPEUTICS DAKO DENMARK A/S (DK) 2009-04-02 WO disclosed