SCHEMBL19851081

SCHEMBL19851081

c1ccc(CCNc2nc(-c3ccc(-c4cccc(CCNc5nc(-c6cccnc6)cs5)c4)cc3)cs2)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.83
RAB9A P51151 6/20 0.83
NPC1 O15118 6/20 0.83
MAPT P10636 5/20 0.83
SMN1; SMN2 Q16637 4/20 0.83
KDM4E B2RXH2 1/20 0.67
GAA P10253 1/20 0.67
HTT P42858 1/20 0.67
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2D6 P10635 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
MEN1 O00255 5/20 0.57
KMT2A Q03164 5/20 0.57
POLB P06746 1/20 0.57
ROCK2 O75116 2/20 0.56
AURKB Q96GD4 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.52
ROCK1 Q13464 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19851055 0.91 RAB9A (1.00) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL205954 0.85 ALDH1A1 (0.84) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL205694 0.85 RAB9A (0.76) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL12297576 0.85 GAA (0.82) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL19850997 0.84 RAB9A (0.59) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
Fanetizole SCHEMBL1813401 0.82 GAA (0.86) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL206058 0.82 RAB9A (0.81) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
Fanetizole SCHEMBL11365554 0.81 GAA (0.84) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL27754680 0.81 MAPT (0.79) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL206769 0.79 ALDH1A1 (0.90) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018027193-A1 GP130 MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-02-08 WO disclosed