SCHEMBL19852053

SCHEMBL19852053

COC(=O)C1=CC=NC(C)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.35
LMNA P02545 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
THRB P10828 1/20 0.34
CHRM1 P11229 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
BLM P54132 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
PTPN1 P18031 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 3/20 0.31
TSHR P16473 1/20 0.31
GABRR1 P24046 1/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20621483 0.71 CYP2C19 (0.35) TSHRNPC1HPGDRAB9A
SCHEMBL17619517 0.69 SLC6A4 (0.31) NPSR1
SCHEMBL8588994 0.69
SCHEMBL27519680 0.67 PTPN1 (0.39) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL28822133 0.66 CHRM3 (0.43) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL5906945 0.65 PTPN1 (0.50) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL12904771 0.65 TSHR (0.34) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL10064320 0.64 TSHR (0.37) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL13924886 0.64 GABRR1 (0.43) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL19275006 0.64 ALDH1A1 (0.39) CHRM3LMNACHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026371-A1 DUAL NAV1.2/5HT2A INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2018-02-08 WO disclosed