SCHEMBL19852467

SCHEMBL19852467

COc1ccc(-c2ccccc2OC2CCN(CC3Cc4cccnc4C3)CC2)cc1OC1CCN(CC2Cc3ccccc3C2)CC1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 5/20 0.42
HTR2A P28223 3/20 0.41
DRD2 P14416 2/20 0.41
HTR2C P28335 1/20 0.41
PDE4A P27815 4/20 0.40
HTR7 P34969 1/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19852164 0.89 SIGMAR1 (0.44) HTR2ADRD2HTR2CHTR7SIGMAR1
SCHEMBL21072474 0.81 OPRL1 (0.47) HTR2ADRD2HTR2CHTR7SIGMAR1
SCHEMBL19852349 0.79 SIGMAR1 (0.52) HTR2ADRD2HTR2CHTR7SIGMAR1
SCHEMBL19852154 0.77 OPRK1 (0.44) HTR2AHTR2CHTR7SIGMAR1
SCHEMBL19852464 0.76 GPR6 (0.41) HTR2ADRD2HTR2CHTR7SIGMAR1
SCHEMBL19852013 0.76 SIGMAR1 (0.42) HTR2ADRD2HTR2CHTR7SIGMAR1
SCHEMBL19852159 0.75 PDE10A (0.41) HTR2ADRD2HTR2C
SCHEMBL21071833 0.75 PDE10A (0.41) HTR2ADRD2HTR2C
SCHEMBL19838591 0.74 HTR7 (0.44) HTR2ADRD2HTR2CHTR7SIGMAR1
Hydrochloric Acid SCHEMBL19839881 0.73 HTR7 (0.43) HTR2ADRD2HTR2CHTR7SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026371-A1 DUAL NAV1.2/5HT2A INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2018-02-08 WO disclosed