SCHEMBL19853660

SCHEMBL19853660

O=C(CCO)N[C@@H](COCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.52
FOLH1 Q04609 1/20 0.51
MBTPS1 Q14703 1/20 0.46
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
CTSL P07711 1/20 0.45
PPARA Q07869 1/20 0.44
TACR1 P25103 2/20 0.44
MMP9 P14780 1/20 0.44
MMP14 P50281 1/20 0.44
MME P08473 1/20 0.43
POLB P06746 1/20 0.43
KLK7 P49862 1/20 0.42
KLK5 Q9Y337 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3365762 0.89 ACE (0.52) ACEFOLH1MBTPS1CTSSCTSK
Hydrochloric Acid SCHEMBL3365449 0.88 ACE (0.51) ACEFOLH1MBTPS1CTSSCTSK
SCHEMBL20804457 0.80 PPARA (0.53) FOLH1CTSSCTSKCTSLPPARA
SCHEMBL20804450 0.77 FOLH1 (0.49) FOLH1CTSSCTSKCTSLPPARA
SCHEMBL28517232 0.77 FAAH (0.50)
SCHEMBL28517231 0.77 FAAH (0.50)
SCHEMBL7518373 0.76 PPARA (0.74) ACECTSSCTSKCTSLPPARA
SCHEMBL19853661 0.76 PPARA (0.74) ACECTSSCTSKCTSLPPARA
SCHEMBL7523142 0.76 ACE (0.50) ACEFOLH1CTSSCTSKCTSL
SCHEMBL1170973 0.76 CTSK (0.56) FOLH1CTSSCTSKCTSLPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026763-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed