SCHEMBL19853781

SCHEMBL19853781

COc1ccc(CN2CC3(CCC(NO)CC3)C2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.50
MMP13 P45452 1/20 0.50
GAA P10253 1/20 0.45
GRM2 Q14416 1/20 0.44
LMNA P02545 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HDAC6 Q9UBN7 2/20 0.42
HDAC1 Q13547 2/20 0.42
CYP3A4 P08684 1/20 0.42
OPRM1 P35372 4/20 0.41
OPRL1 P41146 4/20 0.41
CMA1 P23946 1/20 0.41
MCHR1 Q99705 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RIPK1 Q13546 1/20 0.41
HDAC3 O15379 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19839346 0.86 GAA (0.48) MMP1MMP13GAAGRM2LMNA
SCHEMBL19839918 0.85 GAA (0.49) MMP1MMP13GAAGRM2OPRM1
SCHEMBL19853665 0.84 GAA (0.48) MMP1MMP13GAAGRM2OPRM1
SCHEMBL19853779 0.82 GAA (0.51) MMP1MMP13GAAGRM2OPRM1
SCHEMBL19853780 0.81 MEN1 (0.46) OPRM1OPRL1MEN1KMT2ARIPK1
SCHEMBL19839342 0.77 RIPK1 (0.46) OPRM1OPRL1MEN1KMT2ARIPK1
SCHEMBL24634171 0.75 GAA (0.45) MMP1MMP13GAAGRM2HDAC6
SCHEMBL19853782 0.74 RIPK1 (0.51) GAAOPRM1OPRL1MEN1KMT2A
SCHEMBL17761442 0.74 HDAC1 (0.54) GAALMNASMN1; SMN2HDAC6HDAC1
Nevadistinel SCHEMBL19838866 0.73 GAA (0.51) MMP1MMP13GAAGRM2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026763-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed