SCHEMBL19853780

SCHEMBL19853780

COc1ccc(CN2CC3(CCC(NOCc4ccccc4)CC3)C2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
OPRM1 P35372 12/20 0.43
OPRL1 P41146 12/20 0.43
RIPK1 Q13546 1/20 0.43
SIGMAR1 Q99720 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19839342 0.84 RIPK1 (0.46) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL19853782 0.82 RIPK1 (0.51) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL19853781 0.81 MMP1 (0.50) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL19839918 0.78 GAA (0.49) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL19853665 0.77 GAA (0.48) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL19839346 0.77 GAA (0.48) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL19853779 0.76 GAA (0.51) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL18982937 0.71 NPC1 (0.43) SIGMAR1
SCHEMBL30801694 0.70 OPRM1 (0.39) MEN1KMT2AOPRM1OPRL1RIPK1
SCHEMBL28425659 0.70 SPHK1 (0.49) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026763-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed