SCHEMBL19856858

SCHEMBL19856858

CC(C)(C)C(NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)Cc1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.39
CYP51A1 Q16850 3/20 0.38
MCHR1 Q99705 1/20 0.38
DRD3 P35462 5/20 0.37
HTR2C P28335 3/20 0.37
HTR1A P08908 2/20 0.37
HTR2A P28223 2/20 0.37
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
PYGL P06737 2/20 0.36
PYGM P11217 1/20 0.36
CCKBR P32239 1/20 0.36
STAT6 P42226 1/20 0.36
ESR1 P03372 1/20 0.35
CTNNB1 P35222 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19856857 1.00 DRD2 (0.39) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL19856948 0.88 DRD2 (0.38) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL19856946 0.88 DRD2 (0.38) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL4050168 0.87 DRD2 (0.36) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL19856911 0.86 ESR1 (0.40) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL19856912 0.86 ESR1 (0.40) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL4055536 0.86 DRD2 (0.35) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL4059685 0.85 MCHR1 (0.39) DRD2CYP51A1MCHR1DRD3PYGL
SCHEMBL4058360 0.83 DRD2 (0.36) DRD2CYP51A1MCHR1DRD3HTR2C
SCHEMBL4058066 0.83 MMP2 (0.36) DRD2CYP51A1MCHR1DRD3HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925857-B1 USE OF TRPV4 ANTAGONISTS TO AMELIORATE HYDROCEPHALUS AND RELATED MATERIALS AND METHODS UNIV INDIANA RES & TECH CORP (US) 2018-02-14 EP claimed