SCHEMBL19856946

SCHEMBL19856946

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)c1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.38
MCHR1 Q99705 1/20 0.37
CYP51A1 Q16850 3/20 0.37
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
CRHR1 P34998 3/20 0.37
PYGL P06737 3/20 0.37
PYGM P11217 1/20 0.37
STAT6 P42226 1/20 0.36
HTR2C P28335 2/20 0.36
DRD3 P35462 2/20 0.36
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36
ESR1 P03372 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
CCKAR P32238 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19856948 1.00 DRD2 (0.38) DRD2MCHR1CYP51A1HCRTR1HCRTR2
SCHEMBL19856912 0.94 ESR1 (0.40) DRD2MCHR1CYP51A1PYGLPYGM
SCHEMBL19856911 0.94 ESR1 (0.40) DRD2MCHR1CYP51A1PYGLPYGM
SCHEMBL19856917 0.91 HCRTR1 (0.36) DRD2MCHR1CYP51A1HCRTR1HCRTR2
SCHEMBL19856896 0.91 PYGL (0.43) DRD2CYP51A1PYGLSTAT6DRD3
SCHEMBL19856898 0.91 PYGL (0.43) DRD2CYP51A1PYGLSTAT6DRD3
SCHEMBL19856942 0.90 DRD2 (0.42) DRD2CYP51A1PYGLSTAT6HTR2C
SCHEMBL19856943 0.90 DRD2 (0.42) DRD2CYP51A1PYGLSTAT6HTR2C
SCHEMBL1549871 0.88 CYP51A1 (0.40) DRD2CYP51A1PYGLSTAT6CCKAR
SCHEMBL19856858 0.88 DRD2 (0.39) DRD2MCHR1CYP51A1PYGLPYGM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925857-B1 USE OF TRPV4 ANTAGONISTS TO AMELIORATE HYDROCEPHALUS AND RELATED MATERIALS AND METHODS UNIV INDIANA RES & TECH CORP (US) 2018-02-14 EP claimed