SCHEMBL19859615

SCHEMBL19859615

CON(C)C(=O)c1cc(OCc2ccccc2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.46
ALOX5 P09917 2/20 0.45
NR4A2 P43354 1/20 0.45
APP P05067 1/20 0.45
LTB4R Q15722 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.44
KMT2A Q03164 2/20 0.44
P4HTM Q9NXG6 1/20 0.44
MEN1 O00255 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
CYP2D6 P10635 1/20 0.43
LNPEP Q9UIQ6 1/20 0.43
SRD5A2 P31213 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20510001 0.81 LMNA (0.52) MAOBNR4A2KMT2AP4HTMMEN1
SCHEMBL11617562 0.81 P4HTM (0.60) MAOBALOX5NR4A2KMT2AP4HTM
SCHEMBL3735815 0.81 CLK1 (0.48) KMT2AMEN1KDM4EALDH1A1PKM
SCHEMBL569919 0.81 P4HTM (0.66) MAOBALOX5NR4A2LTB4RLTB4R2
SCHEMBL30678236 0.79 MAOB (0.66) MAOBNR4A2KMT2AMEN1SRD5A2
SCHEMBL4200015 0.79 MAOB (0.66) MAOBNR4A2KMT2AMEN1SRD5A2
SCHEMBL23488362 0.78 PARP10 (0.56) MAOBNR4A2KMT2AP4HTMMEN1
SCHEMBL2713772 0.78 CYP2C9 (0.41) KMT2AMEN1KDM4EALDH1A1
SCHEMBL18681644 0.77 CSF1R (0.54) MAOBNR4A2KMT2AP4HTMMEN1
SCHEMBL1034311 0.77 MAOB (0.63) MAOBALOX5NR4A2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3497098-A1 FUMAGILLOL COMPOUNDS AND METHODS OF MAKING AND USING SAME Zafgen, Inc. (US) 2019-06-19 EP disclosed
US-20190169181-A1 FUMAGILLOL COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. 2019-06-06 US disclosed
US-20190169181-A1 FUMAGILLOL COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. 2019-06-06 US disclosed
WO-2018031877-A1 FUMAGILLOL COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. (US) 2018-02-15 WO disclosed
WO-2018031877-A1 FUMAGILLOL COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. (US) 2018-02-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190169181-A1 FUMAGILLOL COMPOUNDS AND METHODS OF MAKING AND USING SAME METAP2, DNPEP, FOLH1 MAOB 275/4885ALOX5 493/4885NR4A2 4636/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.