SCHEMBL4200015

SCHEMBL4200015

CON(C)C(=O)c1cccc(OCc2ccccc2)c1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.66
NR4A2 P43354 5/20 0.65
KMT2A Q03164 3/20 0.63
SMPD1 P17405 1/20 0.59
SRD5A2 P31213 1/20 0.58
PTPN1 P18031 1/20 0.56
MRGPRX4 Q96LA9 1/20 0.54
MEN1 O00255 2/20 0.53
MAOA P21397 1/20 0.53
NR4A1 P22736 1/20 0.52
NR4A3 Q92570 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30678236 1.00 MAOB (0.66) MAOBNR4A2KMT2ASMPD1SRD5A2
SCHEMBL5605259 0.90 SMPD1 (0.65) MAOBNR4A2KMT2ASMPD1MRGPRX4
SCHEMBL5744375 0.88 SLC2A1 (0.54) MAOBNR4A2KMT2ASMPD1MAOA
SCHEMBL5605085 0.88 MAOB (0.68) MAOBNR4A2KMT2ASMPD1MRGPRX4
SCHEMBL5604959 0.86 SMPD1 (0.63) MAOBNR4A2KMT2ASMPD1MAOA
SCHEMBL10466517 0.86 MAOB (0.69) MAOBNR4A2KMT2ASMPD1SRD5A2
SCHEMBL5866349 0.85 GPR132 (0.59)
SCHEMBL25720520 0.85 FFAR1 (0.53) MAOBKMT2ASMPD1MRGPRX4MAOA
SCHEMBL1034311 0.85 MAOB (0.63) MAOBNR4A2KMT2ASRD5A2MEN1
SCHEMBL20103340 0.83 KMT2A (0.49) MAOBNR4A2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12534457-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2026-01-27 US disclosed
US-12528799-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2026-01-20 US disclosed
US-20240317730-A1 HETEROARYL DERIVATIVE COMPOUNDS, AND USES THEREOF VORONOI INC. (KR) 2024-09-26 US disclosed
US-20240262815-A1 HETEROARYL DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT VORONOI INC (KR) 2024-08-08 US disclosed
US-12037330-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2024-07-16 US disclosed
US-12037330-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2024-07-16 US disclosed
US-12037330-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2024-07-16 US disclosed
US-20240166640-A1 HETEROARYL DERIVATIVE COMPOUNDS, AND USES THEREOF VORONOI INC. (KR) 2024-05-23 US disclosed
EP-4342895-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF Voronoi Inc. (KR) 2024-03-27 EP disclosed
EP-4335847-A1 HETEROARYL DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT Voronoi Inc. (KR) 2024-03-13 EP disclosed
US-6946471-B2 2-(2,6-Dichlorophenyl)-Diarylimidazoles HOFFMANN-LA ROCHE INC. (US) 2005-09-20 US disclosed
WO-2005068452-A1 PHENYL-[4-(3-PHENYL-1H-PYRAZOL-4-YL)-PYRIMIDIN-2-YL]-AMINE DERIVATIVES AS IGF-IR INHIBITORS NOVARTIS AG (CH) 2005-07-28 WO disclosed
WO-2005040153-A1 NOVEL TRIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-05-06 WO disclosed
US-20050085473-A1 Novel triarylimidazoles HOFFMANN-LA ROCHE INC. 2005-04-21 US disclosed
EP-1499577-A1 2-(2,6-DICHLOROPHENYL)-DIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-01-26 EP disclosed
US-20040214874-A1 2-(2,6-Dichlorophenyl)-Diarylimidazoles BRANDT MICHAEL 2004-10-28 US disclosed
US-6790852-B2 HETEROCYCLIC NITROGEN COMPOUNDS SUCH AS 2-(2,6-DICHLOROPHENYL) -4-(3-BROMOPHENYL)-5-(2-(3- HYDROXYPROPYLAMINO)PYRIMIDIN-4-YL) -N-H-IMIDAZOLE, USED AS TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC OR ANTITUMOR AGENTS HOFFMANN-LA ROCHE INC. 2004-09-14 US disclosed
US-20030199691-A1 2-(2,6-dichlorophenyl)-diarylimidazoles F. HOFFMANN-LA ROCHE AG (CH) 2003-10-23 US disclosed
WO-2003087026-A1 2-(2,6-DICHLOROPHENYL)-DIARYLIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2003-10-23 WO disclosed
WO-2002022584-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085473-A1 Novel triarylimidazoles AURKAIP1, GLS2, GOT2 MAOB 1708/4885NR4A2 1677/4885KMT2A 2396/4885
US-12037330-B2 Heteroaryl derivative compounds, and uses thereof ERBB2, EGFR, ERBB3 MAOB 1885/4885NR4A2 1988/4885KMT2A 2221/4885
US-20030199691-A1 2-(2,6-dichlorophenyl)-diarylimidazoles CYP2D6, CYP2F1, CYP1A2 MAOB 414/4885NR4A2 2261/4885KMT2A 933/4885
US-20240262815-A1 HETEROARYL DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT ERBB2, ERBB4, ERBB3 MAOB 3672/4885NR4A2 152/4885KMT2A 990/4885
US-20240317730-A1 HETEROARYL DERIVATIVE COMPOUNDS, AND USES THEREOF ERBB2, EGFR, ERBB3 MAOB 1885/4885NR4A2 1988/4885KMT2A 2221/4885
US-12528799-B2 Heteroaryl derivative compounds, and uses thereof ERBB2, EGFR, ERBB3 MAOB 3077/4885NR4A2 267/4885KMT2A 2396/4885
US-20040214874-A1 2-(2,6-Dichlorophenyl)-Diarylimidazoles CYP2D6, CYP1A2, CYP2F1 MAOB 476/4885NR4A2 2155/4885KMT2A 858/4885
US-12534457-B2 Heteroaryl derivative compounds, and uses thereof ERBB2, EGFR, ERBB3 MAOB 2014/4885NR4A2 2421/4885KMT2A 2771/4885
US-20240166640-A1 HETEROARYL DERIVATIVE COMPOUNDS, AND USES THEREOF ERBB2, EGFR, ERBB3 MAOB 1885/4885NR4A2 1988/4885KMT2A 2221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.