SCHEMBL19860025

SCHEMBL19860025

Cc1c(F)cc(F)cc1-c1c[nH]c2ncc(-c3cnn(S(=O)(=O)N4CCN(C)CC4)c3)cc12

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIK1 P57059 1/20 0.46
SIK3 Q9Y2K2 1/20 0.46
ALK Q9UM73 10/20 0.45
MAP4K1 Q92918 1/20 0.44
TNIK Q9UKE5 4/20 0.43
PDPK1 O15530 3/20 0.40
MAP3K11 Q16584 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15805270 0.89 SIK1 (0.59) SIK1SIK3ALKMAP4K1TNIK
SCHEMBL19860027 0.80 SIK1 (0.65) SIK1SIK3ALKTNIKPDPK1
SCHEMBL19860023 0.78 SIK1 (0.60) SIK1SIK3ALKMAP4K1TNIK
SCHEMBL19860026 0.77 SIK1 (0.59) SIK1SIK3ALKTNIKPDPK1
SCHEMBL15805266 0.77 MAP4K1 (0.49) MAP4K1TNIKMAP3K11
SCHEMBL17636867 0.77 SIK1 (0.43) SIK1SIK3ALKMAP4K1TNIK
SCHEMBL21677080 0.76 MAP4K1 (0.48) MAP4K1TNIKMAP3K11
SCHEMBL19860022 0.73 SIK1 (0.79) SIK1SIK3ALKPDPK1
SCHEMBL19860029 0.71 SIK1 (0.35) SIK1SIK3ALKMAP4K1
SCHEMBL15799467 0.69 SIK1 (0.82) SIK1SIK3ALKMAP4K1TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890153-B2 Substituted 1H-pyrrolo [2, 3-b] pyridine and 1H-pyrazolo [3, 4-b] pyridine derivatives as salt inducible kinase 2 (SIK2) inhibitors ARRIEN PHARMACEUTICALS LLC (US) 2018-02-13 US disclosed