SCHEMBL19873652

SCHEMBL19873652

CC(OC(=O)Nc1cc(Cl)sc1-c1ccc(-c2ccc(C3CC3)cc2)nc1)c1ccsc1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 1/20 0.36
LPAR3 Q9UBY5 1/20 0.36
DGAT1 O75907 7/20 0.33
NAAA Q02083 1/20 0.32
CDK13 Q14004 1/20 0.30
IDO1 P14902 1/20 0.30
ENPP2 Q13822 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19873634 0.90 LPAR1 (0.38) LPAR1LPAR3NAAAENPP2
SCHEMBL19873601 0.90 LPAR1 (0.38) LPAR1LPAR3NAAAENPP2
SCHEMBL19873636 0.89 LPAR1 (0.46) LPAR1LPAR3DGAT1NAAA
SCHEMBL19873635 0.89 LPAR1 (0.46) LPAR1LPAR3DGAT1NAAA
SCHEMBL28387786 0.88 MEN1 (0.31)
SCHEMBL19873626 0.87 DGAT1 (0.33) LPAR1LPAR3DGAT1IDO1ENPP2
SCHEMBL17367451 0.86 LPAR1 (0.36) LPAR1LPAR3
SCHEMBL17215491 0.86 LPAR1 (0.42) LPAR1LPAR3
SCHEMBL19873555 0.84 LPAR1 (0.34) LPAR1LPAR3NAAA
SCHEMBL19873553 0.84 LPAR1 (0.34) LPAR1LPAR3NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3360869-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND USEFUL FOR THE TREATMENT OF DISEASES CAUSED BY LPA. UBE INDUSTRIES (JP) 2020-07-29 EP claimed
EP-2940013-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND UBE INDUSTRIES (JP) 2018-02-21 EP claimed