SCHEMBL19873660

SCHEMBL19873660

C[C@@H](OC(=O)Nc1cc(F)sc1-c1ccc(-c2ccc(C3CC3)cc2)cc1)c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 1/20 0.39
LPAR3 Q9UBY5 1/20 0.39
NAAA Q02083 1/20 0.39
CCR1 P32246 3/20 0.36
FFAR2 O15552 2/20 0.36
CHRM3 P20309 5/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
APP P05067 1/20 0.34
IDO1 P14902 1/20 0.34
PRCP P42785 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19873662 1.00 LPAR1 (0.39) LPAR1LPAR3NAAACCR1FFAR2
SCHEMBL22260989 0.92 LPAR1 (0.40) LPAR1LPAR3NAAACHRM3CHRM2
SCHEMBL22260988 0.92 LPAR1 (0.40) LPAR1LPAR3NAAACHRM3CHRM2
SCHEMBL19873665 0.91 NAAA (0.41) LPAR1LPAR3NAAACCR1IDO1
SCHEMBL19873663 0.91 NAAA (0.41) LPAR1LPAR3NAAACCR1IDO1
SCHEMBL19873608 0.91 APP (0.38) LPAR1LPAR3NAAACCR1CHRM3
SCHEMBL19873606 0.91 APP (0.38) LPAR1LPAR3NAAACCR1CHRM3
SCHEMBL19873617 0.90 LPAR1 (0.48) LPAR1LPAR3NAAAAPP
SCHEMBL19873618 0.90 LPAR1 (0.48) LPAR1LPAR3NAAAAPP
SCHEMBL19873574 0.90 CHRM3 (0.37) LPAR1LPAR3NAAACCR1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3360869-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND USEFUL FOR THE TREATMENT OF DISEASES CAUSED BY LPA. UBE INDUSTRIES (JP) 2020-07-29 EP claimed
EP-2940013-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND UBE INDUSTRIES (JP) 2018-02-21 EP claimed