SCHEMBL19890263

SCHEMBL19890263

CCOC(=O)C1(O)CNC(c2ccccc2)=N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.44
BRD4 O60885 1/20 0.43
OPRM1 P35372 5/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
OPRD1 P41143 3/20 0.39
OPRK1 P41145 3/20 0.39
SLC22A1 O15245 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23027868 0.70 GABRA2 (0.41) OPRM1SMN1; SMN2RAB9ANPC1CYP1A2
SCHEMBL835869 0.69 OPRM1 (0.57) BRD4OPRM1SMN1; SMN2OPRD1OPRK1
SCHEMBL830705 0.69 OPRM1 (0.57) BRD4OPRM1SMN1; SMN2OPRD1OPRK1
SCHEMBL17051307 0.68 SMN1; SMN2 (0.48) ATMBRD4OPRM1SMN1; SMN2RAB9A
SCHEMBL13036615 0.67 ALDH1A1 (0.41) ATMSMN1; SMN2CYP1A2CYP2C19ALDH1A1
SCHEMBL9416753 0.66 ALDH1A1 (0.49) OPRM1SMN1; SMN2RAB9ANPC1CYP1A2
SCHEMBL28788636 0.66 SMN1; SMN2 (0.46) OPRM1SMN1; SMN2RAB9ANPC1CYP1A2
SCHEMBL6315068 0.65 OPRM1 (0.40) BRD4OPRM1SMN1; SMN2RAB9ANPC1
SCHEMBL25401575 0.65 ITGB1 (0.48) ATMBRD4OPRM1SMN1; SMN2RAB9A
SCHEMBL6401268 0.65 OPRM1 (0.40) BRD4OPRM1SMN1; SMN2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018033642-A1 HETEROCYCLIC LIPXON ANALOGS AND USES THEROF UNIVERSITY COLLEGE DUBLIN (IE) 2018-02-22 WO disclosed