SCHEMBL19901352

SCHEMBL19901352

CC(C)(C)NC(=O)c1cc2cc(N)ccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.51
CYP2A6 P11509 1/20 0.46
KEAP1 Q14145 1/20 0.46
HDAC2 Q92769 1/20 0.46
KDM4E B2RXH2 3/20 0.45
GAA P10253 2/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44
TP53 P04637 2/20 0.44
POLB P06746 1/20 0.44
PYGL P06737 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
PIN1 Q13526 1/20 0.42
PLD2 O14939 1/20 0.41
PLD1 Q13393 1/20 0.41
ABL1 P00519 1/20 0.41
PDGFRB P09619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14845703 0.84 PIN1 (0.62) HRH4HDAC2KDM4EGAAALDH1A1
SCHEMBL12501351 0.83 ALOX15 (0.55) HRH4CYP2A6KEAP1HDAC2KDM4E
SCHEMBL25782820 0.82 F7 (0.60) HRH4KMT2APYGLNPC1RAB9A
SCHEMBL13334344 0.82 TP53 (0.47) HRH4KDM4EGAAKMT2AALDH1A1
SCHEMBL12669766 0.80 KDM4E (0.64) KDM4EGAAALDH1A1MAPK1NPC1
SCHEMBL12392310 0.80 HRH4 (0.55) HRH4CYP2A6KEAP1KDM4EALDH1A1
SCHEMBL12826973 0.80 KDM4E (0.64) KDM4EGAAKMT2AALDH1A1PYGL
SCHEMBL12848263 0.79 ALOX15 (0.58) HRH4CYP2A6KEAP1HDAC2KDM4E
SCHEMBL12862877 0.78 HRH4 (0.58) HRH4CYP2A6KEAP1HDAC2KDM4E
SCHEMBL1415238 0.77 KDM4E (0.61) HRH4HDAC2KDM4EALDH1A1PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9901567-B2 Substituted CC-1065 analogs and their conjugates SYNTARGA B.V. (NL) 2018-02-27 US disclosed