SCHEMBL19902709

SCHEMBL19902709

O=C(N[C@H]1CC[C@H](c2n[nH]c(=O)c3ccccc32)CC1)c1ccc(N2CCCC2)cn1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.50
PRKAA2 P54646 1/20 0.46
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 1/20 0.44
ACKR3 P25106 2/20 0.43
MGLL Q99685 1/20 0.42
WNT1 P04628 1/20 0.40
DYRK1A Q13627 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17452954 0.88 ROCK2 (0.58) PARP1PRKAA2ROCK2ROCK1ACKR3
SCHEMBL20229924 0.81 ROCK2 (0.43) PRKAA2ROCK2ROCK1
SCHEMBL19902507 0.81 DHODH (0.42) ROCK2ROCK1ACKR3
SCHEMBL19902565 0.80 USP30 (0.47) ROCK2ROCK1WNT1DYRK1A
SCHEMBL19902356 0.80 CHRNA7 (0.45) PARP1ROCK2ROCK1
SCHEMBL19902716 0.79 USP30 (0.51) ROCK2ROCK1DYRK1A
SCHEMBL19902631 0.77 HDAC8 (0.42) PARP1ROCK2ROCK1
SCHEMBL27390382 0.76 PARP1 (0.48) PARP1
SCHEMBL19902343 0.75 ALDH1A1 (0.43) PARP1ROCK2ROCK1
SCHEMBL30944627 0.75 PARP1 (0.46) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed