SCHEMBL19904646

SCHEMBL19904646

O=C[C@H]1CCN(c2ccc3c(c2)CCCC3)C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.41
TSHR P16473 1/20 0.37
KDM2B Q8NHM5 3/20 0.36
AVPR2 P30518 1/20 0.35
HCAR1 Q9BXC0 1/20 0.35
CYP17A1 P05093 1/20 0.34
NOTUM Q6P988 1/20 0.34
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
TMEM97 Q5BJF2 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
AR P10275 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16695240 0.75 NOTUM (0.62) NOTUM
SCHEMBL16695146 0.74 NOTUM (0.47) HTR6KDM2BNOTUMSMN1; SMN2
SCHEMBL16684690 0.74 NOTUM (0.47) HTR6KDM2BNOTUMSMN1; SMN2
SCHEMBL16695100 0.74 NOTUM (0.47) HTR6KDM2BNOTUMSMN1; SMN2
SCHEMBL21704260 0.73 HRH4 (0.53)
Hydrochloric Acid SCHEMBL17913779 0.73 ESR1 (0.48) KDM2BTMEM97SIGMAR1
SCHEMBL26099884 0.73 TRIM24 (0.38) NOTUMTRIM24TRIM33ALDH1A1KDM4E
SCHEMBL26099880 0.73 TRIM24 (0.38) NOTUMTRIM24TRIM33ALDH1A1KDM4E
SCHEMBL19904404 0.73 GHSR (0.42) TRIM24MAOB
SCHEMBL5691206 0.73 IP6K1 (0.48) HTR6TSHRHCAR1CYP17A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed