SCHEMBL19905481

SCHEMBL19905481

CNC(=O)c1ncnc2c(C(C)[C@H](C)CNc3cc(-c4ccc(OC)nc4)ncn3)cccc12

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.40
FAAH O00519 6/20 0.38
HDAC1 Q13547 9/20 0.36
PIK3CA P42336 8/20 0.36
USP2 O75604 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17874673 0.92 PRKDC (0.46) PRKDCFAAHHDAC1PIK3CAUSP2
SCHEMBL19905441 0.91 PRKDC (0.44) PRKDCFAAHUSP2CYP1A2CYP3A4
SCHEMBL19905491 0.89 PRKDC (0.44) PRKDCFAAH
SCHEMBL19905365 0.89 PRKDC (0.41) PRKDCFAAH
SCHEMBL19905199 0.88 PRKDC (0.38) PRKDCFAAHHDAC1PIK3CAUSP2
SCHEMBL19905448 0.88 FAAH (0.47) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL19905258 0.83 PRKDC (0.37) PRKDCFAAH
SCHEMBL17874675 0.83 PRKDC (0.50) PRKDCFAAHUSP2CYP1A2CYP3A4
SCHEMBL15473153 0.83 PRKDC (0.50) PRKDCFAAHUSP2CYP1A2CYP3A4
SCHEMBL19355626 0.83 PRKDC (0.44) PRKDCFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed