SCHEMBL19905441

SCHEMBL19905441

CNC(=O)c1ncnc2c(C(C)[C@H](C)CNc3cc(-c4cnc(OC)nc4)ncn3)cccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.44
FAAH O00519 10/20 0.38
CYP1A2 P05177 5/20 0.33
CYP3A4 P08684 5/20 0.33
CYP2D6 P10635 5/20 0.33
CLK4 Q9HAZ1 5/20 0.33
CYP2C19 P33261 4/20 0.33
TSHR P16473 3/20 0.33
HSD17B10 Q99714 3/20 0.33
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33
TP53 P04637 2/20 0.33
MAPK1 P28482 2/20 0.33
HIF1A Q16665 2/20 0.33
USP2 O75604 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ALOX15 P16050 2/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905491 0.94 PRKDC (0.44) PRKDCFAAHTP53ABL1BCR
SCHEMBL15473153 0.92 PRKDC (0.50) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL17874675 0.92 PRKDC (0.50) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL19905481 0.91 PRKDC (0.40) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL19905365 0.88 PRKDC (0.41) PRKDCFAAH
SCHEMBL19905459 0.87 PRKDC (0.42) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL19905448 0.86 FAAH (0.47) PRKDCFAAHCYP1A2CYP3A4CYP2D6
SCHEMBL17874683 0.86 PRKDC (0.51) PRKDCFAAHTP53ABL1BCR
SCHEMBL19905088 0.83 PRKDC (0.48) PRKDCFAAHTP53ABL1BCR
SCHEMBL17874673 0.83 PRKDC (0.46) PRKDCFAAHCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed