SCHEMBL19905940

SCHEMBL19905940

Cc1cc2[nH]ncc2cc1-c1cc(-c2nc3cc(C)c(CC(=O)O)c(-c4ccc(Cl)cc4OC(C)(C)C)c3s2)ccn1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
STK17B O94768 1/20 0.32
MAP3K8 P41279 1/20 0.32
STK17A Q9UEE5 1/20 0.32
SHMT1 P34896 1/20 0.32
MAPK8 P45983 1/20 0.31
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
ROCK1 Q13464 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905899 0.90 CCNE1 (0.33) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19905941 0.88 PTGDR2 (0.39) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906069 0.84 EGFR (0.35) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906229 0.84 EIF4E (0.36) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906268 0.84 EIF4E (0.38) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906239 0.83 PTGDR2 (0.35) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906288 0.83 CSF1R (0.35) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906328 0.83 PTGER1 (0.34) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906369 0.83 KDM4E (0.38) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906211 0.83 KDM4E (0.34) KDM4EMEN1ALDH1A1KMT2APTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed