SCHEMBL19906080

SCHEMBL19906080

Cc1cc2nc(-c3ccnc(-c4ccc5c(c4)c(C4CC4)nn5C)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.35
CACNA1H O95180 1/20 0.33
PTGDR2 Q9Y5Y4 6/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE5A O76074 1/20 0.31
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE7A Q13946 1/20 0.31
PDE1C Q14123 1/20 0.31
PDE3A Q14432 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
BRD4 O60885 3/20 0.31
CREBBP Q92793 3/20 0.31
FABP4 P15090 1/20 0.31
FABP5 Q01469 1/20 0.31
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906076 0.90 KDM4E (0.37) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL19906078 0.90 SHMT1 (0.31) CNR1PTGDR2KDM4EMEN1ALDH1A1
SCHEMBL20030418 0.89 CNR1 (0.39) CNR1CACNA1HPTGDR2KDM4EMEN1
SCHEMBL19906043 0.88 SLC2A1 (0.36) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL20030905 0.86 KDM4E (0.35) CNR1PTGDR2KDM4EMEN1ALDH1A1
SCHEMBL20030967 0.85 CNR1 (0.37) CNR1PTGDR2KDM4EMEN1ALDH1A1
SCHEMBL20030655 0.85 CNR1 (0.36) CNR1PTGDR2KDM4EMEN1ALDH1A1
SCHEMBL20030730 0.85 CNR1 (0.36) CNR1PTGDR2KDM4EMEN1ALDH1A1
SCHEMBL15341104 0.84 CYP3A4 (0.36) CNR1CACNA1H
SCHEMBL19905816 0.84 KDM4E (0.35) PTGDR2KDM4EMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed