SCHEMBL19906147

SCHEMBL19906147

Cc1cc2nc(-c3ccc4c(c3)c(C(C)C)nn4C)sc2c(-c2ccc(Cl)cc2OC(C)(C)C)c1CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
S1PR1 P21453 1/20 0.32
HSD17B10 Q99714 1/20 0.31
AKR1B1 P15121 1/20 0.31
SHMT1 P34896 1/20 0.31
CPT1A P50416 1/20 0.31
CPT1B Q92523 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
MAPK8 P45983 1/20 0.31
PDE5A O76074 1/20 0.30
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE4D Q08499 1/20 0.30
PDE7A Q13946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905856 0.90 KDM4E (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906148 0.88 PTGDR2 (0.39) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906280 0.86 KDM4E (0.34) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906171 0.85 KDM4E (0.36) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906167 0.84 PTGES2 (0.36) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906192 0.84 PTGDR2 (0.32) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906405 0.84 KDM4E (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906379 0.83 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906197 0.83 PTGDR2 (0.36) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906078 0.82 SHMT1 (0.31) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed