SCHEMBL19908457

SCHEMBL19908457

Cc1cnc2c(c1)N(C(=O)c1ccccc1)CCN2

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.48
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CRBN Q96SW2 2/20 0.40
GRM5 P41594 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 2/20 0.39
STAT3 P40763 1/20 0.39
HTT P42858 1/20 0.39
ALK Q9UM73 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GPR6 P46095 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1601376 0.85 NOS1 (0.48) NOS1ALDH1A1HPGDRAB9AKMT2A
SCHEMBL19908281 0.82 ALDH1A1 (0.45) ALDH1A1RAB9ASMN1; SMN2GRM5HSD17B10
SCHEMBL1601639 0.80 NOS1 (0.53) NOS1ALDH1A1HPGDNPC1RAB9A
SCHEMBL1600998 0.80 AVPR2 (0.49) NOS1POLBSTAT3ALKHSD17B10
SCHEMBL3601421 0.80 NOS1 (0.49) NOS1ALDH1A1HPGDCRBNALK
SCHEMBL3601417 0.79 ALK (0.49) NOS1ALK
SCHEMBL1601622 0.79 ALK (0.47) NOS1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL1601053 0.78 POLB (0.55) ALDH1A1NPC1GRM5POLBALK
SCHEMBL14387373 0.78 ALK (0.38) ALDH1A1ALKGPR6
SCHEMBL1601615 0.73 CAMK2D (0.46) HPGDALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091951-B1 PYRIDO[2,3-B]PYRAZINE AND [1,8]-NAPHTHYRIDINE DERIVATIVES AS ALK AND C-MET INHIBITORS CEPHALON INC (US) 2018-02-28 EP disclosed