SCHEMBL1990893

SCHEMBL1990893

CS(=O)(Cc1csc(C(F)(F)F)n1)=NC#N

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.32
CDK9 P50750 1/20 0.32
MCHR1 Q99705 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7601458 0.80 KMT2A (0.40)
SCHEMBL3084435 0.79 SLC6A3 (0.33) CDK2CDK9
SCHEMBL20530847 0.73 MCHR1 (0.33) MCHR1
SCHEMBL305535 0.73 CDK2 (0.34) CDK2CDK9
SCHEMBL6923900 0.70 MAPT (0.33) MCHR1
SCHEMBL9262966 0.67 MCHR1 (0.34) MCHR1
SCHEMBL24415623 0.65 HRH1 (0.40)
SCHEMBL119494 0.65 CDK2 (0.39) CDK2CDK9
SCHEMBL17263328 0.65 CCR4 (0.40) MCHR1
SCHEMBL21205449 0.64 CDK2 (0.33) CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2338885-B1 Insecticidal N-Substituted (2-Substituted-1,3-Thiazol) Alkyl Sulfoximines DOW AGROSCIENCES LLC (US) 2012-10-31 EP disclosed
EP-2338885-B1 Insecticidal N-Substituted (2-Substituted-1,3-Thiazol) Alkyl Sulfoximines DOW AGROSCIENCES LLC (US) 2012-10-31 EP disclosed
EP-2057135-B1 INSECTICIDAL N-SUBSTITUTED (2- SUBSTITUTED-1,3-THIAZOL) ALKYL SULFOXIMINES DOW AGROSCIENCES LLC (US) 2012-06-13 EP disclosed
EP-2057135-B1 INSECTICIDAL N-SUBSTITUTED (2- SUBSTITUTED-1,3-THIAZOL) ALKYL SULFOXIMINES DOW AGROSCIENCES LLC (US) 2012-06-13 EP disclosed
US-8183270-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES, LLC (US) 2012-05-22 US disclosed
US-8183270-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES, LLC (US) 2012-05-22 US disclosed
EP-2338883-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338883-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338885-A1 Insecticidal N-Substituted (2-Substituted-1,3-Thiazol) Alkyl Sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338884-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338884-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
US-20110060018-A1 INSECTICIDAL N-SUBSTITUTED (2-SUBSTITUTED-1,3-THIAZOL)ALKYL SULFOXIMINES CORTEVA AGRISCIENCE LLC 2011-03-10 US disclosed
US-20110060018-A1 INSECTICIDAL N-SUBSTITUTED (2-SUBSTITUTED-1,3-THIAZOL)ALKYL SULFOXIMINES CORTEVA AGRISCIENCE LLC 2011-03-10 US disclosed
US-7863303-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2011-01-04 US disclosed
US-7863303-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2011-01-04 US disclosed
US-7863303-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2011-01-04 US disclosed
WO-2008027539-A1 INSECTICIDAL N-SUBSTITUTED (2- SUDSTITUTED-1,3-THIAZOL) ALKYL SULFOXIMINES DOW AGROSCIENCES LLC (US) 2008-03-06 WO disclosed
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2008-03-06 US disclosed
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2008-03-06 US disclosed
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2008-03-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines TST, NIT2, MSL1 CDK2 2909/4885CDK9 4413/4885MCHR1 2202/4885
US-20110060018-A1 INSECTICIDAL N-SUBSTITUTED (2-SUBSTITUTED-1,3-THIAZOL)ALKYL SULFOXIMINES TST, NIT2, MSL1 CDK2 2909/4885CDK9 4413/4885MCHR1 2202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.