SCHEMBL19910474

SCHEMBL19910474

O=Cc1ccc(CNCc2cncc(F)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.41
LMNA P02545 1/20 0.39
NAMPT P43490 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ALDH1A1 P00352 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADORA2B P29275 1/20 0.36
KMT2A Q03164 1/20 0.36
PDPK1 O15530 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12640358 0.80 CYP2C9 (0.43) NAMPTCYP2C9HDAC1ALDH1A1ADORA2B
SCHEMBL4054709 0.79 LMNA (0.59) LMNACYP2C9ALDH1A1KMT2ACYP2D6
SCHEMBL2599996 0.78 ADORA2B (0.41) NAMPTCYP2C9ALDH1A1ADORA2BPDPK1
SCHEMBL16709818 0.76 LMNA (0.49) LMNANAMPTALDH1A1KMT2AKDM4E
SCHEMBL12675604 0.74 PDPK1 (0.38) NOS1NAMPTCYP2C9CYP11B1CYP11B2
SCHEMBL17568760 0.73 NOS1 (0.41) NOS1LMNANAMPTCYP2C9CYP11B1
SCHEMBL12640370 0.72 PDPK1 (0.37) NOS1NAMPTCYP2C9ALDH1A1ADORA2B
SCHEMBL30775165 0.71 NAMPT (0.45) NOS1NAMPTCYP2C9CYP11B1CYP11B2
SCHEMBL10483931 0.70 NOS1 (0.51) NOS1NAMPTCYP2C9CYP11B1CYP11B2
SCHEMBL7981783 0.70 NOS1 (0.45) NOS1NAMPTCYP2C9CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3065738-B1 COMPOSITIONS AND METHODS FOR MODULATING FARNESOID X RECEPTORS NOVARTIS AG (CH) 2018-02-28 EP disclosed