SCHEMBL19918909

SCHEMBL19918909

C=C(C)Cc1cc(F)c(C2CCCCC2)cc1CC

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
JAK3 P52333 1/20 0.34
PTGDR2 Q9Y5Y4 3/20 0.33
NUDT1 P36639 1/20 0.31
BACE1 P56817 1/20 0.31
PTGDR Q13258 1/20 0.31
HTR2A P28223 2/20 0.31
CAMKK1 Q8N5S9 1/20 0.30
CAMKK2 Q96RR4 1/20 0.30
EPHX2 P34913 1/20 0.30
DPP4 P27487 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24962101 0.79 NUDT1 (0.42) JAK2JAK1JAK3PTGDR2NUDT1
SCHEMBL8264162 0.71 OPRL1 (0.38) SCN9A
SCHEMBL2748088 0.68 HTR2A (0.39) NUDT1BACE1HTR2AEPHX2DPP4
SCHEMBL11702604 0.66 NUDT1 (0.44) JAK2JAK1JAK3PTGDR2NUDT1
SCHEMBL23441849 0.66 OPRL1 (0.39) PTGDR2NUDT1BACE1PTGDR
SCHEMBL12354267 0.66 CHRNB2 (0.40) PTGDR2NUDT1BACE1PTGDRHTR2A
SCHEMBL11366020 0.65 NUDT1 (0.43) PTGDR2NUDT1BACE1
SCHEMBL14314452 0.65 NUDT1 (0.46) JAK2JAK1JAK3PTGDR2NUDT1
SCHEMBL16014088 0.65 NUDT1 (0.45) PTGDR2NUDT1BACE1PTGDR
SCHEMBL10776428 0.64 NUDT1 (0.42) JAK2JAK1JAK3PTGDR2NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367800-B1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF DISEASES SUCH AS CANCER BOEHRINGER INGELHEIM INT (DE) 2018-02-28 EP disclosed