SCHEMBL19920890

SCHEMBL19920890

[CH]1CNC(c2ccncn2)=N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 2/20 0.36
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CDK9 P50750 2/20 0.36
CCNA1 P78396 2/20 0.36
CDK5 Q00535 2/20 0.36
CDK5R1 Q15078 2/20 0.36
CDC7 O00311 1/20 0.35
HSP90AA1 P07900 1/20 0.34
MAPK14 Q16539 2/20 0.34
MAPK9 P45984 2/20 0.34
MAPK13 O15264 1/20 0.34
RAF1 P04049 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
CYP2D6 P10635 1/20 0.33
MAPK10 P53779 1/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
CDC42BPB Q9Y5S2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30595872 0.71 HSP90AA1 (0.52) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL2814353 0.71 HSP90AA1 (0.52) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL27612098 0.69 NISCH (0.59) CYP2D6
SCHEMBL13910999 0.69 HSP90AA1 (0.50) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL10402322 0.67 HSP90AA1 (0.48) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL19814593 0.66
SCHEMBL9903935 0.65 CYP2D6 (0.60) HSP90AA1MAPK14MAPK9MAPK13RAF1
SCHEMBL27995610 0.64 LATS1 (0.33) CDC7HSP90AA1MAPK14MAPK9MAPK13
SCHEMBL4789542 0.63 SIGMAR1 (0.47) CDC7
SCHEMBL25295479 0.63 TP53 (0.48) CCNT1CCNA2CDK2CDK9CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3289876-A1 COMPOUNDS FOR TREATMENT OF CANCER University of Tennessee Research Foundation (US) 2018-03-07 EP disclosed