SCHEMBL27612098

SCHEMBL27612098

c1cc(C2=NCCN2)ncn1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 13/20 0.59
CYP1A2 P05177 3/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
ALOX15 P16050 1/20 0.45
LMNA P02545 2/20 0.44
PMP22 Q01453 1/20 0.44
RECQL P46063 1/20 0.42
TOP2A P11388 1/20 0.41
TOP2B Q02880 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30373758 0.74 NISCH (1.00) NISCHCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL1345182 0.74 NISCH (1.00) NISCHCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL548286 0.73 NISCH (0.55) NISCHCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL10507263 0.71 NISCH (1.00) NISCHLMNARECQLTOP2ATOP2B
SCHEMBL30595872 0.71 HSP90AA1 (0.52) CYP1A2KDM4ECYP2D6LMNA
SCHEMBL2814353 0.71 HSP90AA1 (0.52) CYP1A2KDM4ECYP2D6LMNA
SCHEMBL4110363 0.71 NISCH (1.00) NISCHCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL4726421 0.70 NISCH (0.56) NISCHCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL19920890 0.69 CCNT1 (0.36) CYP2D6
SCHEMBL13910999 0.69 HSP90AA1 (0.50) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1829509-A Pharmaceutical composition for treating tumors COMBINATORX INC (US) 2006-09-06 CN claimed
CN-1681511-A Combinations of drugs for the treatment of neoplasms COMBINATORX INC (US) 2005-10-12 CN claimed
CN-1878556-A Combinations of drugs for the treatment of neoplasms COMBINATORX INC (US) 2006-12-13 CN disclosed
CN-1681511-A Combinations of drugs for the treatment of neoplasms COMBINATORX INC (US) 2005-10-12 CN disclosed