SCHEMBL1992607

SCHEMBL1992607

O=S1(=O)N[C]c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA9 Q16790 4/20 0.38
CA4 P22748 3/20 0.38
CA7 P43166 3/20 0.38
KDM4E B2RXH2 3/20 0.38
KMT2A Q03164 2/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
BCHE P06276 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
MEN1 O00255 1/20 0.37
NOX1 Q9Y5S8 1/20 0.37
GPR3 P46089 1/20 0.36
HTT P42858 1/20 0.33
KEAP1 Q14145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9983691 0.70 CA12 (0.35) CA12CA1CA2CA9CA4
SCHEMBL3714644 0.65 CA12 (0.35) CA12CA1CA2CA9CA4
SCHEMBL1947435 0.64 CA12 (0.34) CA12CA1CA2CA9CA4
SCHEMBL29374033 0.64 CA12 (0.46) CA12CA1CA2CA9CA4
SCHEMBL2563736 0.64 CA12 (0.46) CA12CA1CA2CA9CA4
SCHEMBL9551845 0.62 GPR3 (0.39) CA12CA1CA2CA9CA4
SCHEMBL6228752 0.62 GPR3 (0.39) CA12CA1CA2CA9CA4
SCHEMBL1450925 0.60 GPR3 (0.37) CA12CA1CA2CA9CA4
SCHEMBL5485319 0.60 GPR3 (0.37) CA12CA1CA2CA9CA4
SCHEMBL8336188 0.60 CA12 (0.64) CA12CA1CA2CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344494-B1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS SIGNAL PHARM LLC (US) 2016-04-20 EP claimed
US-8299056-B2 Aminotriazolopyridines, compositions thereof, and methods of treatment therewith SIGNAL PHARMACEUTICALS, LLC (US) 2012-10-30 US claimed
EP-2344494-A1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS Signal Pharmaceuticals, LLC (US) 2011-07-20 EP claimed
US-20100093698-A1 AMINOTRIAZOLOPYRIDINES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC 2010-04-15 US claimed
WO-2010027500-A1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2010-03-11 WO claimed
US-10131646-B2 Aromatic sulfonium salt compound, photoacid generator, resist composition, cationic polymerization initiator, and cationically polymerizable composition ADEKA CORPORATION (JP) 2018-11-20 US disclosed
US-20180079738-A1 AROMATIC SULFONIUM SALT COMPOUND, PHOTOACID GENERATOR, RESIST COMPOSITION, CATIONIC POLYMERIZATION INITIATOR, AND CATIONICALLY POLYMERIZABLE COMPOSITION ADEKA CORPORATION (JP) 2018-03-22 US disclosed
EP-3272744-A1 AROMATIC SULFONIUM SALT COMPOUND, PHOTOACID GENERATOR, RESIST COMPOSITION, CATIONIC POLYMERIZATION INITIATOR, AND CATIONICALLY POLYMERIZABLE COMPOSITION Adeka Corporation (JP) 2018-01-24 EP disclosed
EP-2344494-B1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS SIGNAL PHARM LLC (US) 2016-04-20 EP disclosed
US-9073854-B2 Aromatic sulfonium salt compound ADEKA CORPORATION (JP) 2015-07-07 US disclosed
EP-2502915-B1 AROMATIC SULFONIUM SALT COMPOUND ADEKA CORP (JP) 2015-03-18 EP disclosed
US-20130005707-A1 AMINOTRIAZOLOPYRIDINES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BAHMANYAR SOGOLE (US) 2013-01-03 US disclosed
WO-2010027500-A1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2010-03-11 WO disclosed
EP-1109071-A1 2-(1,2-benzisothiazol-3(2h)-ylidene 1,1-dioxide)acetamides negative charge control agents for electrostatographic toners and developers EASTMAN KODAK COMPANY (US) 2001-06-20 EP disclosed
US-6184387-B1 2-(1,2-benzisothiazol-3(2H)-ylidene 1,1-dioxide)acetamides negative charge control agents for electrostatographic toners and developers EASTMAN KODAK COMPANY 2001-02-06 US disclosed
US-6165668-A N-[2-(1,2-benzisothiazol-3(2H)-ylidene 1,1-dioxide)-2-cyanoacetyl]benzenesulfonamide charge control agents for electrostatographic toners and developers EASTMAN KODAK COMPANY (US) 2000-12-26 US disclosed
US-6120964-A TONERS WITH BINDERS EASTMAN KODAK COMPANY (US) 2000-09-19 US disclosed
US-5849450-A (1,2-benzisothiazol-3-(2H)-ylidene 1,1-dioxide) acetate-terminated polymer charge-control agents for electrostatographic toners and developers EASTMAN KODAK COMPANY (US) 1998-12-15 US disclosed
US-5744277-A Electrostatographic toners and developers containing (1,2-benzisothiazol-3-(2H)-ylidene 1,1-dioxide) acetate-terminated polymer charge-control agents EASTMAN KODAK COMPANY (US) 1998-04-28 US disclosed
US-5723248-A Electrostatographic toners and developers containing bis 1,2-benzisthiazol-3(2h) -ylidene 1,1-dioxide) acetates!charge-control agents EASTMAN KODAK COMPANY (US) 1998-03-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130005707-A1 AMINOTRIAZOLOPYRIDINES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH MAP3K2, MAP3K1, MAP3K3 CA12 4880/4885CA1 4826/4885CA2 4075/4885
US-10131646-B2 Aromatic sulfonium salt compound, photoacid generator, resist composition, cationic polymerization initiator, and cationically polymerizable composition ASIC1, NOX5, SLC6A19 CA12 231/4885CA1 166/4885CA2 21/4885
US-20100093698-A1 AMINOTRIAZOLOPYRIDINES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH MAP3K2, MAP3K1, MAP3K3 CA12 4880/4885CA1 4826/4885CA2 4075/4885
US-20180079738-A1 AROMATIC SULFONIUM SALT COMPOUND, PHOTOACID GENERATOR, RESIST COMPOSITION, CATIONIC POLYMERIZATION INITIATOR, AND CATIONICALLY POLYMERIZABLE COMPOSITION ASIC1, NOX5, SLC6A19 CA12 231/4885CA1 166/4885CA2 21/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.