SCHEMBL19936552

SCHEMBL19936552

CCNc1ccc(CO)cc1C=N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
RECQL P46063 1/20 0.35
IDO1 P14902 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
GFER P55789 1/20 0.34
PLEC Q15149 1/20 0.34
EGFR P00533 1/20 0.34
HCAR3 P49019 1/20 0.31
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
ERN1 O75460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19936608 0.87 CYP3A4 (0.35) CYP3A4TSHRRECQLIDO1KDM4E
SCHEMBL22073753 0.77 ALDH1A1 (0.38) CYP3A4TSHRRECQLIDO1KDM4E
SCHEMBL21317742 0.76 STAT3 (0.42) CYP3A4TSHRRECQLIDO1KDM4E
SCHEMBL19936583 0.74 ALDH1A1 (0.60) KDM4EALDH1A1GAAMAPTTHRB
SCHEMBL16976666 0.74 KDM4E (0.56) CYP3A4TSHRRECQLIDO1KDM4E
SCHEMBL14402733 0.71 CNR1 (0.38) TSHRKDM4EALDH1A1GAAMAPT
SCHEMBL19707177 0.71 IDO1 (0.40) CYP3A4TSHRRECQLIDO1KDM4E
SCHEMBL26473856 0.70 TRPA1 (0.39) KDM4EALDH1A1GAAMAPTHTT
SCHEMBL28201373 0.70 ALDH1A1 (0.37) CYP3A4TSHRRECQLIDO1KDM4E
SCHEMBL23642619 0.70 MAPT (0.50) CYP3A4KDM4EALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2594555-B1 HETEROCYCLIC COMPOUND, AND p27 KIP1 DEGRADATION INHIBITOR ASKA PHARM CO LTD (JP) 2018-03-07 EP disclosed