SCHEMBL19936600

SCHEMBL19936600

CNc1sc(-c2ccc(Cl)cc2C)nc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.40
NOTUM Q6P988 2/20 0.39
APP P05067 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
RAB9A P51151 3/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 2/20 0.36
POLB P06746 2/20 0.36
ESR1 P03372 1/20 0.36
CRHR1 P34998 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
SHMT1 P34896 1/20 0.34
SHMT2 P34897 1/20 0.34
NOX1 Q9Y5S8 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
AGPAT2 O15120 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19936434 0.84 MAPT (0.37) APPSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL14960175 0.83 CASP3 (0.41) CASP3NOTUMSMN1; SMN2RAB9AMAPT
SCHEMBL19936424 0.82 HSP90AA1 (0.46) MAPTNPC1POLBCRHR1KDM4E
SCHEMBL19936382 0.81 HDAC9 (0.39) APPMAPT
SCHEMBL2069606 0.77 SMN1; SMN2 (0.56) CASP3APPSMN1; SMN2RAB9AMAPT
SCHEMBL3436690 0.76 KDM4E (0.42) CASP3NOTUMSMN1; SMN2RAB9AMAPT
SCHEMBL19936529 0.76 HSD11B1 (0.40) APPSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL5548627 0.76 NOTUM (0.38) CASP3NOTUMSMN1; SMN2RAB9AMAPT
SCHEMBL3436648 0.75 KDM4E (0.65) CASP3SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL14800709 0.74 GAA (0.68) SMN1; SMN2RAB9AMAPTNPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2594555-B1 HETEROCYCLIC COMPOUND, AND p27 KIP1 DEGRADATION INHIBITOR ASKA PHARM CO LTD (JP) 2018-03-07 EP disclosed