SCHEMBL19937643

SCHEMBL19937643

Nc1ncc(-c2ccn(C3CCC3)n2)cc1C1CC1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 18/20 0.50
INSR P06213 1/20 0.41
NPM1 P06748 1/20 0.41
ALK Q9UM73 1/20 0.41
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR3 P22607 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19937663 0.97 MAP3K12 (0.50) MAP3K12INSRNPM1ALK
SCHEMBL19937610 0.83 MAP3K12 (0.51) MAP3K12INSRNPM1ALK
SCHEMBL19937757 0.81 MAP3K12 (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937642 0.80 MAP3K12 (0.55) MAP3K12
SCHEMBL19937622 0.80 MAP3K12 (0.52) MAP3K12INSRNPM1ALKFGFR1
SCHEMBL19937609 0.80 INSR (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937864 0.79 MAP3K12 (0.52) MAP3K12FGFR1FGFR2FGFR3
SCHEMBL19937789 0.79 INSR (0.42) MAP3K12INSRNPM1ALKFGFR1
SCHEMBL19937751 0.78 MAP3K12 (0.53) MAP3K12
SCHEMBL19937634 0.78 MAP3K11 (0.52) MAP3K12INSRNPM1ALKFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945938-B1 3-SUBSTITUTED PYRAZOLES AND USE AS DLK INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-07 EP disclosed